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Bretazenil CAS#84379-13-5

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Chemical Name：Bretazenil

CAS No.84379-13-5

Molecular Formula：C19H20BrN3O3

Molecular weight:418.28

Sample: Available

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Product Details

Products Description of Bretazenil CAS#84379-13-5

Brotacetin is a partial agonist of the GABAA receptor of the benzodiazepine class. It was first developed by Roche as an antianxiety drug. Studies have found that brotacetin can counteract the spasms caused by pentamethazine. At an antispasmodic dose (125-250 μg·kg-1), brotacetin combined with pyridostigmine (100 μg·kg-1, im) and aprofen (4 mg·kg-1, im) can prevent sarin and soman poisoning. Brotacetin has good antianxiety activity at a dose of 50-400 μg·kg-1. Compared with diazepam, it has little adverse reaction of myasthenia. Therefore, as one of the components for protecting the central nervous system, it has obvious advantages.

Bretazenil Chemical Properties

Boiling point	594.3±50.0 °C(Predicted)
density	1.56±0.1 g/cm3(Predicted)
storage temp.	2-8°C
solubility	DMSO: 24 mg/mL, soluble
form	solid
pka	0.78±0.20(Predicted)
color	white
InChI	InChI=1S/C19H20BrN3O3/c1-19(2,3)26-18(25)15-16-13-8-5-9-22(13)17(24)14-11(20)6-4-7-12(14)23(16)10-21-15/h4,6-7,10,13H,5,8-9H2,1-3H3/t13-/m0/s1
InChIKey	LWUDDYHYYNNIQI-ZDUSSCGKSA-N
SMILES	N12C=NC(C(OC(C)(C)C)=O)=C1[C@]1([H])CCCN1C(=O)C1=C(Br)C=CC=C12